SCHEMBL878121

SCHEMBL878121

C=CCOC(=O)CN(C)C(=O)Cc1ccccc1Oc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.47
HTR2A P28223 4/20 0.47
SLC6A2 P23975 4/20 0.47
SLC6A3 Q01959 4/20 0.47
SLC1A5 Q15758 1/20 0.42
PPARA Q07869 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.37
CHRM1 P11229 1/20 0.37
MAPT P10636 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
KCNH2 Q12809 2/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
CCR8 P51685 1/20 0.35
TSPO P30536 1/20 0.35
CXCL8 P10145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9995320 0.88 SLC6A4 (0.52) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5
SCHEMBL872624 0.85 SLC6A4 (0.53) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5
SCHEMBL8471261 0.80 SLC6A4 (0.58) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5
SCHEMBL12361548 0.79 SLC6A4 (0.54) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5
SCHEMBL13474499 0.76 SLC6A4 (0.53) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5
SCHEMBL11648424 0.76 SMN1; SMN2 (0.45) SLC6A4SLC6A2PPARAMEN1KMT2A
SCHEMBL12353135 0.75 SLC6A4 (0.50) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5
SCHEMBL14636285 0.75 NPSR1 (0.44) SLC6A4SLC6A2SLC6A3POLBCHRM1
SCHEMBL1146416 0.75 HTR2A (0.54) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5
SCHEMBL28801696 0.73 PPARA (0.54) SLC6A4HTR2ASLC6A2SLC6A3SLC1A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038975-A2 PROCESS FOR THE PREPARATION OF (3ARS,12BRS)-5-CHLORO-2-METHYL-2,3,3A12B-TETRAHYDRO-1HDIBENZO[2,3:6,7] OXEPINO [4,5-C]PYRROLE MALEATE AND IT'S PHARMACEUTICAL COMPOSITION THEREOF MSN LABORATORIES LIMITED (IN) 2012-03-29 WO claimed
WO-2012038975-A2 PROCESS FOR THE PREPARATION OF (3ARS,12BRS)-5-CHLORO-2-METHYL-2,3,3A12B-TETRAHYDRO-1HDIBENZO[2,3:6,7] OXEPINO [4,5-C]PYRROLE MALEATE AND IT'S PHARMACEUTICAL COMPOSITION THEREOF MSN LABORATORIES LIMITED (IN) 2012-03-29 WO disclosed