SCHEMBL8782001

SCHEMBL8782001

Cc1cccc(Nc2ncnc3ccc(-c4nc5ccccc5[nH]4)cc23)c1

nearest known ligand 0.74

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.74
MET P08581 11/20 0.74
EGFR P00533 3/20 0.62
HTT P42858 1/20 0.61
HIF1A Q16665 1/20 0.61
ERBB2 P04626 2/20 0.58
MAPK1 P28482 1/20 0.58
CD38 P28907 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8782234 0.82 EGFR (0.62) KDRMETEGFRHTTHIF1A
SCHEMBL6187944 0.81 BRAF (0.73) EGFRHTTHIF1AERBB2MAPK1
SCHEMBL4355660 0.79 EGFR (0.55) KDRMETEGFRHTTHIF1A
SCHEMBL3391554 0.78 EGFR (1.00) KDREGFRHTTHIF1AERBB2
SCHEMBL8871863 0.78 EGFR (0.82) EGFRHTTHIF1AERBB2MAPK1
SCHEMBL13620922 0.77 EGFR (0.67) EGFRHTTHIF1AERBB2MAPK1
SCHEMBL159209 0.75 EGFR (1.00) EGFRHTTHIF1AERBB2MAPK1
SCHEMBL29350058 0.75 EGFR (1.00) EGFRHTTHIF1AERBB2MAPK1
SCHEMBL4349199 0.75 MAPK1 (1.00) EGFRHTTHIF1AERBB2MAPK1
SCHEMBL6884208 0.74 KDR (0.49) KDRMETEGFRHTTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0794953-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1997-09-17 EP disclosed
WO-1996016960-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1996-06-06 WO disclosed