SCHEMBL8784389

SCHEMBL8784389

CN1CCC(c2c[nH]c3ccc(Cc4nc[nH]n4)cc23)C1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
ATM Q13315 1/20 0.54
HTR1D P28221 9/20 0.52
HTR1B P28222 9/20 0.52
HTR1A P08908 2/20 0.52
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
THPO P40225 1/20 0.49
NOS3 P29474 2/20 0.47
NOS1 P29475 2/20 0.47
GABRP O00591 1/20 0.47
GABRD O14764 1/20 0.47
GABRA1 P14867 1/20 0.47
GABRB1 P18505 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8784576 0.94 HTR1D (0.59) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL8784390 0.82 HTR1D (0.53) KDM4EATMHTR1DHTR1BHTR1A
SCHEMBL8508032 0.82 KDM4E (0.64) KDM4EATMHTR1DHTR1BHTR1A
SCHEMBL9269516 0.81 KDM4E (0.62) KDM4EATMHTR1DHTR1BHTR1A
SCHEMBL9268538 0.77 HTR1D (0.71) KDM4EATMHTR1DHTR1BHTR1A
SCHEMBL8784342 0.76 HTR1A (0.53) KDM4EATMHTR1DHTR1BHTR1A
Hydrochloric Acid SCHEMBL9269587 0.76 HTR1D (0.57) KDM4EATMHTR1DHTR1BHTR1A
SCHEMBL8508491 0.75 KDM4E (0.68) KDM4EATMHTR1DHTR1BHTR1A
SCHEMBL8784644 0.75 HTR1D (0.53) KDM4EATMHTR1DHTR1BHTR1A
SCHEMBL9272206 0.75 HTR1D (0.88) KDM4EATMHTR1DHTR1BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497512-B1 Imidazole, triazole and tetrazole derivatives MERCK SHARP & DOHME (GB) 1997-09-24 EP claimed