SCHEMBL8784402

SCHEMBL8784402

COc1ccc(COCc2c(-c3ccccc3)c3cc(C)c(C)cc3c(=O)n2C)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.55
KCNH2 Q12809 1/20 0.55
TACR1 P25103 12/20 0.55
F2RL3 Q96RI0 1/20 0.47
DPP4 P27487 4/20 0.42
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPK8 P45983 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8785109 0.91 TACR1 (0.61) KCNA5KCNH2TACR1F2RL3DPP4
SCHEMBL8785635 0.85 TACR1 (0.61) KCNA5KCNH2TACR1F2RL3DPP4
SCHEMBL3115349 0.84 KCNA5 (0.76) KCNA5KCNH2TACR1F2RL3DPP4
SCHEMBL8785202 0.83 TACR1 (0.72) KCNA5KCNH2TACR1F2RL3DPP4
SCHEMBL1379988 0.82 KCNA5 (0.64) KCNA5KCNH2TACR1F2RL3DPP4
Hydrochloric Acid SCHEMBL3112400 0.81 KCNA5 (0.62) KCNA5KCNH2TACR1F2RL3DPP4
SCHEMBL8785655 0.80 TACR1 (0.56) KCNA5KCNH2TACR1KDM4ESMN1; SMN2
SCHEMBL8785588 0.78 TACR1 (0.68) KCNA5KCNH2TACR1F2RL3DPP4
SCHEMBL1382996 0.77 KCNA5 (0.76) KCNA5KCNH2TACR1F2RL3DPP4
SCHEMBL8786372 0.77 TACR1 (0.51) KCNA5KCNH2TACR1F2RL3DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585913-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-12-29 EP disclosed
US-5700810-A Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-23 US disclosed
US-5482967-A LOWERING CHOLESTEROL TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-01-09 US disclosed
EP-0585913-A2 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-09 EP disclosed