SCHEMBL878556

SCHEMBL878556

CCOC(=O)c1cc2c(cc1F)C(N)CC2

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
ACHE P22303 7/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
LMNA P02545 1/20 0.40
JMJD6 Q6NYC1 1/20 0.40
TSHR P16473 2/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL803251 0.85 ACHE (0.42) ACHETSHR
Hydrochloric Acid SCHEMBL785262 0.83 ACHE (0.44) ACHETSHR
Hydrochloric Acid SCHEMBL785261 0.83 ACHE (0.44) ACHETSHR
SCHEMBL803162 0.79 ACHE (0.42) KDM4EACHETSHR
SCHEMBL803167 0.78 ACHE (0.40) KDM4EACHEAKR1C3AKR1C2
SCHEMBL877871 0.78 ACHE (0.40) KDM4EACHEAKR1C3AKR1C2
Hydrochloric Acid SCHEMBL484838 0.78 ACHE (0.44) ACHETSHR
Hydrochloric Acid SCHEMBL484839 0.78 ACHE (0.44) ACHETSHR
Hydrochloric Acid SCHEMBL785346 0.77 ACHE (0.42) KDM4EACHEAKR1C3AKR1C2
Hydrochloric Acid SCHEMBL785269 0.77 ACHE (0.42) KDM4EACHEAKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed