SCHEMBL878739

SCHEMBL878739

c1ccc(COCc2nc(-c3ccnc4c3CCN4)no2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
RAB9A P51151 9/20 0.38
NPC1 O15118 8/20 0.38
SMN1; SMN2 Q16637 6/20 0.38
MAPK1 P28482 4/20 0.38
TDP1 Q9NUW8 4/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
ALDH1A1 P00352 3/20 0.37
S1PR1 P21453 2/20 0.36
S1PR3 Q99500 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
MAPT P10636 4/20 0.35
TSHR P16473 3/20 0.35
CASP3 P42574 2/20 0.35
SENP8 Q96LD8 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12959974 0.76 MAPT (0.50) RAB9ANPC1SMN1; SMN2MAPK1TDP1
SCHEMBL858200 0.75 S1PR1 (0.48) RAB9ANPC1SMN1; SMN2MAPK1TDP1
SCHEMBL13138653 0.70 S1PR1 (0.39) RAB9ANPC1SMN1; SMN2ALDH1A1S1PR1
SCHEMBL14441202 0.64 TDP1 (0.51) RAB9ANPC1SMN1; SMN2MAPK1TDP1
SCHEMBL12346375 0.63 MRGPRX4 (0.31)
SCHEMBL6691870 0.61 TSHR (0.54) RAB9ANPC1SMN1; SMN2MAPK1TDP1
SCHEMBL13138769 0.61 PARP1 (0.45) ALDH1A1TSHRKDM4EHPGDHSD17B10
SCHEMBL858129 0.61 RAB9A (0.55) RAB9ANPC1SMN1; SMN2MAPK1TDP1
SCHEMBL858331 0.60 NPC1 (0.52) RAB9ANPC1SMN1; SMN2TDP1L3MBTL1
SCHEMBL9491202 0.59 TSHR (0.94) ALDH1A1TSHRKDM4ELMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143271-B2 Compounds and methods for kinase modulation, and indications therefor PLEXXIKON INC. (US) 2012-03-27 US disclosed