SCHEMBL8788249

SCHEMBL8788249

ClCCC1COc2ccccc2O1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.61
CA2 P00918 3/20 0.55
ADRA2A P08913 2/20 0.53
ADRA1A P35348 2/20 0.53
HTR1A P08908 2/20 0.53
DRD1 P21728 1/20 0.53
TBXA2R P21731 1/20 0.53
SLC6A2 P23975 1/20 0.53
DRD3 P35462 1/20 0.53
ADRA2B P18089 1/20 0.53
ADRA2C P18825 1/20 0.53
ADRA1D P25100 1/20 0.53
ADRA1B P35368 1/20 0.53
SCN1A P35498 1/20 0.53
SCN2A Q99250 1/20 0.53
SCN3A Q9NY46 1/20 0.53
SIGMAR1 Q99720 1/20 0.51
POLB P06746 2/20 0.50
ESR2 Q92731 1/20 0.50
MTNR1A P48039 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2204596 0.85 ADRA2A (0.56) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL1568393 0.81 HTT (0.66) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL1545537 0.81 HTT (0.66) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL406531 0.81 HTT (0.61) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL5871673 0.81 HTT (0.61) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL12309752 0.81 POLB (0.62) HTTCA2ADRA2AADRA1AHTR1A
Hydrochloric Acid SCHEMBL8179101 0.80 HTT (0.59) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL11238168 0.80 HTT (0.59) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL10978442 0.79 HTT (0.58) HTTCA2ADRA2AADRA1AHTR1A
SCHEMBL12602022 0.79 POLB (0.59) HTTCA2ADRA2AADRA1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0395244-B1 Pyridine derivatives WYETH JOHN & BROTHER LTD (GB) 1997-02-19 EP disclosed
US-5194439-A 5-HT Agonists or Antagonists, Nervous System Disorders, Hypotensive Agents JOHN WYETH & BROTHER LIMITED (GB) 1993-03-16 US disclosed
US-5075303-A Central nervous system disorders JOHN WYETH & BROTHER LIMITED (GB) 1991-12-24 US disclosed
EP-0395244-A1 Pyridine derivatives JOHN WYETH & BROTHER LIMITED (GB) 1990-10-31 EP disclosed