SCHEMBL8790874

SCHEMBL8790874

[CH2]CC(=O)C1CCCc2ccccc2N1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
SMYD3 Q9H7B4 1/20 0.45
MTNR1A P48039 3/20 0.43
MME P08473 8/20 0.40
ACE P12821 4/20 0.39
HTR1A P08908 2/20 0.38
HTR2A P28223 2/20 0.38
DRD3 P35462 2/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP1A2 P05177 1/20 0.38
F2 P00734 1/20 0.37
F10 P00742 1/20 0.37
PLG P00747 1/20 0.37
PRSS1 P07477 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8791310 0.84 MAPT (0.50) MAPTGAASMYD3MTNR1AMME
SCHEMBL17675115 0.83 MAPT (0.65) MAPTGAASMYD3MTNR1AMME
SCHEMBL32680077 0.81 MAPT (0.50) MAPTGAASMYD3MTNR1AMME
SCHEMBL8067762 0.81 MAPT (0.50) MAPTGAASMYD3MTNR1AMME
SCHEMBL4734530 0.77 SMYD3 (0.56) MAPTGAASMYD3MTNR1AHTR1A
SCHEMBL1545216 0.77 SMYD3 (0.52) MAPTGAASMYD3MTNR1AHTR1A
SCHEMBL4730904 0.77 SMYD3 (0.52) MAPTGAASMYD3MTNR1AHTR1A
SCHEMBL8401235 0.75 MAPT (0.48) MAPTGAASMYD3MTNR1AMME
SCHEMBL17647218 0.74 MAPT (0.47) MAPTGAASMYD3MTNR1AMME
SCHEMBL4019694 0.74 SMYD3 (0.58) MAPTGAASMYD3MTNR1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560235-B1 Condensed heterocyclic ketone derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-06-04 EP disclosed
US-5462934-A Cholinesterase inhibitor; learning enhancement TAKEDA CHEMICAL INDUSTRIES (JP) 1995-10-31 US disclosed
EP-0560235-A1 Condensed heterocyclic ketone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-09-15 EP disclosed