SCHEMBL8797368

SCHEMBL8797368

CC(C)c1cccc(C(C)C)c1NC(=O)C1c2ccccc2COc2ccc(CO)cc21

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.38
LMNA P02545 2/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SOAT1 P35610 3/20 0.37
SOAT2 O75908 2/20 0.37
MEN1 O00255 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
TBXAS1 P24557 1/20 0.36
S1PR4 O95977 1/20 0.35
S1PR5 Q9H228 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797055 0.92 TP53 (0.38) TP53LMNAKMT2ASMN1; SMN2SOAT1
SCHEMBL8797272 0.86 TP53 (0.45) TP53LMNAKMT2ASMN1; SMN2
SCHEMBL8798173 0.86 TP53 (0.47) TP53LMNAKMT2ASMN1; SMN2MEN1
SCHEMBL8797541 0.85 LPAR1 (0.45) TP53LMNAKMT2ASMN1; SMN2MEN1
SCHEMBL8797024 0.85 GRM7 (0.41) TP53LMNAKMT2ASMN1; SMN2MEN1
SCHEMBL8797451 0.85 TP53 (0.39) TP53LMNAKMT2ASMN1; SMN2SOAT1
SCHEMBL8797482 0.85 LPAR1 (0.45) TP53LMNAKMT2ASMN1; SMN2SOAT1
SCHEMBL8797584 0.84 TBXAS1 (0.48) LMNAKMT2ATBXAS1
SCHEMBL8797835 0.84 TP53 (0.38) TP53LMNAKMT2ASMN1; SMN2SOAT1
SCHEMBL8797398 0.84 LPAR1 (0.49) TP53LMNAKMT2ASMN1; SMN2SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0497201-B1 Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO KK (JP) 1997-01-15 EP disclosed
US-5478835-A Acyl coenzyme A: acyltransferase inhibitors; treatment of hyperlipemia and arteriosclerosis KYOWA HAKKO KOGYO CO., LTD. (JP) 1995-12-26 US disclosed
US-5340807-A Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-08-23 US disclosed
EP-0497201-A1 Tricyclic compounds and intermediates thereof KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-08-05 EP disclosed