SCHEMBL8797441

SCHEMBL8797441

Cc1cc(C)nc(NC(=O)CN)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.63
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
LMNA P02545 3/20 0.57
LCK P06239 1/20 0.54
MAPT P10636 2/20 0.52
CHRNB2 P17787 1/20 0.52
CHRNB4 P30926 1/20 0.52
CHRNA3 P32297 1/20 0.52
CHRNA4 P43681 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 2/20 0.50
NPC1 O15118 1/20 0.50
GBA1 P04062 1/20 0.50
RAB9A P51151 1/20 0.50
NOS3 P29474 1/20 0.48
NOS2 P35228 1/20 0.48
TP53 P04637 1/20 0.48
SORT1 Q99523 1/20 0.46
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12182431 0.84 MAPK1 (0.65) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL22281653 0.83 MAPK1 (0.63) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL9665242 0.81 MAPK1 (0.70) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL6508707 0.80 KMT2A (0.60) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL9077089 0.80 MAPK1 (0.83) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL8797408 0.80 MAPK1 (0.46) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL30711612 0.80 LCK (0.67) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL4504096 0.80 LCK (0.67) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL50044 0.78 LCK (0.60) MAPK1CYP1A2CYP3A4LMNALCK
SCHEMBL9664290 0.78 MAPK1 (0.74) MAPK1CYP1A2CYP3A4LMNALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0632026-B1 Alpha amino acid derivatives, a method for their preparation and pharmaceutical preparations containing them ADIR (FR) 1997-11-19 EP claimed
US-5470864-A Glycine amide derivatives containing pyridine or pyridine-N-oxide, anticholesterol, antiinflammatory ADIR ET COMPAGNIE (FR) 1995-11-28 US claimed
EP-0632026-B1 Alpha amino acid derivatives, a method for their preparation and pharmaceutical preparations containing them ADIR (FR) 1997-11-19 EP disclosed
US-5585390-A ANTIINFLAMMATORY AGENTS; ANTILIPEMIC AGENTS ADIR ET COMPAGNIE (FR) 1996-12-17 US disclosed
US-5470864-A Glycine amide derivatives containing pyridine or pyridine-N-oxide, anticholesterol, antiinflammatory ADIR ET COMPAGNIE (FR) 1995-11-28 US disclosed
EP-0632026-A1 Alpha amino acid derivatives, a method for their preparation and pharmaceutical preparations containing them ADIR ET COMPAGNIE (FR) 1995-01-04 EP disclosed