SCHEMBL9664290

SCHEMBL9664290

Cc1cc(C)nc(NC(=O)CCCCl)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.74
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
MAPT P10636 3/20 0.51
LMNA P02545 1/20 0.51
LCK P06239 1/20 0.49
CHRNB2 P17787 1/20 0.48
CHRNB4 P30926 1/20 0.48
CHRNA3 P32297 1/20 0.48
CHRNA4 P43681 1/20 0.48
NOS3 P29474 1/20 0.47
NOS2 P35228 1/20 0.47
SMN1; SMN2 Q16637 5/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
ALDH1A1 P00352 3/20 0.46
GBA1 P04062 1/20 0.46
TP53 P04637 1/20 0.44
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9665242 0.83 MAPK1 (0.70) MAPK1CYP1A2CYP3A4MAPTLMNA
SCHEMBL9077089 0.81 MAPK1 (0.83) MAPK1CYP1A2CYP3A4MAPTLMNA
SCHEMBL12182431 0.79 MAPK1 (0.65) MAPK1CYP1A2CYP3A4MAPTLMNA
SCHEMBL9664553 0.79 RAB9A (0.69) MAPTLMNASMN1; SMN2NPC1RAB9A
SCHEMBL20095383 0.79 RAB9A (0.58) MAPTSMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL22281653 0.78 MAPK1 (0.63) MAPK1CYP1A2CYP3A4MAPTLMNA
SCHEMBL8797441 0.78 MAPK1 (0.63) MAPK1CYP1A2CYP3A4MAPTLMNA
SCHEMBL8798095 0.77 MAPK1 (0.70) MAPK1CYP1A2CYP3A4MAPTLMNA
SCHEMBL9080445 0.77 MAPK1 (0.62) MAPK1CYP1A2CYP3A4MAPTLMNA
SCHEMBL8673571 0.76 SMN1; SMN2 (0.52) MAPK1CYP1A2CYP3A4MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519996-A1 IMIDAZOLES RHONE-POULENC RORER LIMITED (GB) 1992-12-30 EP disclosed
WO-1991013876-A1 IMIDAZOLES RHONE-POULENC RORER LIMITED (GB) 1991-09-19 WO disclosed