SCHEMBL8797958

SCHEMBL8797958

Cc1cccc(Nc2cc(NCCOCCO)ncn2)c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.77
TP53 P04637 1/20 0.48
TNNI3K Q59H18 2/20 0.48
KCNH3 Q9ULD8 1/20 0.43
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
GRM1 Q13255 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP6 P55212 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GBA1 P04062 1/20 0.41
HPGD P15428 1/20 0.41
ERBB3 P21860 3/20 0.40
RECQL P46063 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798594 0.85 EGFR (0.85) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL13989431 0.84 EGFR (0.54) EGFRTP53KCNH3NPC1RAB9A
SCHEMBL8799214 0.84 EGFR (0.83) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL27337220 0.81 EGFR (0.78) EGFRTNNI3KNPC1RAB9AMAPT
SCHEMBL1387422 0.81 EGFR (0.65) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL1387302 0.79 EGFR (0.72) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL27408585 0.79 EGFR (0.74) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL7778617 0.77 EGFR (0.64) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL7771252 0.77 EGFR (0.60) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL8317846 0.75 EGFR (0.64) EGFRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed