SCHEMBL8798182

SCHEMBL8798182

CN1Cc2c(-c3ccccc3)cc3[nH]c(=O)c(=O)[nH]c3c2C1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 4/20 0.47
GRIA2 P42262 4/20 0.47
GRIA3 P42263 4/20 0.47
GRIA4 P48058 4/20 0.47
ADORA3 P0DMS8 1/20 0.39
ADORA2B P29275 1/20 0.39
TNKS O95271 1/20 0.39
PARP1 P09874 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14287158 0.90 GRIA1 (0.58) GRIA1GRIA2GRIA3GRIA4
SCHEMBL8537048 0.90 GRIA1 (0.58) GRIA1GRIA2GRIA3GRIA4TNKS
SCHEMBL8533969 0.82 GRIA1 (0.56) GRIA1GRIA2GRIA3GRIA4
SCHEMBL14287157 0.79 GRIA1 (0.46) GRIA1GRIA2GRIA3GRIA4TNKS
SCHEMBL6787042 0.75 GRIA1 (0.52) GRIA1GRIA2GRIA3GRIA4GRIN2D
SCHEMBL6785459 0.75 GRIA1 (0.57) GRIA1GRIA2GRIA3GRIA4
SCHEMBL7103934 0.70 GRIA1 (0.81) GRIA1GRIA2GRIA3GRIA4GRIN2D
SCHEMBL6784941 0.70 GRIA1 (0.48) GRIA1GRIA2GRIA3GRIA4GRIN2D
SCHEMBL6783750 0.70 GRIA1 (0.48) GRIA1GRIA2GRIA3GRIA4
SCHEMBL6783751 0.70 GRIA1 (0.44) GRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0698025-B1 AMPA ANTAGONISTS AND A METHOD OF TREATMENT THEREWITH NEUROSEARCH AS (DK) 1997-12-17 EP disclosed
EP-0538332-B1 POLYCYCLIC GUANINE DERIVATIVES SCHERING CORP (US) 1997-07-23 EP disclosed
US-5393755-A Hypotensive agents, enzyme inhibitors SCHERING CORPORATION (US) 1995-02-28 US disclosed