SCHEMBL8798272

SCHEMBL8798272

Cc1cccc(Nc2cc(NC(CO)CO)ncn2)c1

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.66
TNNI3K Q59H18 4/20 0.53
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HTT P42858 1/20 0.42
HIF1A Q16665 1/20 0.42
THRB P10828 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
ERBB3 P21860 2/20 0.41
MAPT P10636 1/20 0.41
RECQL P46063 1/20 0.41
SYK P43405 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387302 0.84 EGFR (0.72) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL8798355 0.83 EGFR (0.60) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL7771269 0.79 EGFR (0.66) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL2782010 0.78 EGFR (0.65) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL8798594 0.77 EGFR (0.85) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL7777342 0.77 EGFR (0.64) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL8799214 0.76 EGFR (0.83) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL690632 0.76 EGFR (0.62) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL1387422 0.75 EGFR (0.65) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL8798667 0.75 EGFR (0.61) EGFRTNNI3KRAB9AHTTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed