SCHEMBL8798563

SCHEMBL8798563

C=CCNc1cc(Nc2cccc(C)c2)ncn1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.66
TNNI3K Q59H18 4/20 0.53
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
MAPT P10636 2/20 0.44
RECQL P46063 1/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
TP53 P04637 2/20 0.44
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HSD17B10 Q99714 2/20 0.44
JAK3 P52333 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ERBB2 P04626 1/20 0.42
HTT P42858 2/20 0.42
HIF1A Q16665 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387302 0.84 EGFR (0.72) EGFRTNNI3KNPC1RAB9AMEN1
SCHEMBL27337227 0.82 JAK3 (0.50) EGFRTNNI3KNPC1RAB9AJAK3
SCHEMBL27337220 0.81 EGFR (0.78) EGFRTNNI3KNPC1RAB9AMAPT
SCHEMBL17458853 0.81 NPC1 (0.49) EGFRTNNI3KNPC1RAB9AKDM4E
SCHEMBL27408585 0.78 EGFR (0.74) EGFRTNNI3KNPC1RAB9AMAPT
SCHEMBL2782010 0.78 EGFR (0.65) EGFRTNNI3KNPC1RAB9ALMNA
SCHEMBL2857440 0.77 MAPT (0.62) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL8798594 0.77 EGFR (0.85) EGFRTNNI3KNPC1RAB9AMAPT
SCHEMBL8799214 0.76 EGFR (0.83) EGFRTNNI3KNPC1RAB9AMAPT
Hydrochloric Acid SCHEMBL2857434 0.76 MAPT (0.60) NPC1RAB9AMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed