SCHEMBL8798786

SCHEMBL8798786

CC(C)OC(=O)C(C)N1CCc2ccc(N)cc2C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.49
GABRA1 P14867 2/20 0.46
GABRG2 P18507 2/20 0.46
GABRB3 P28472 2/20 0.46
MAPT P10636 5/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 1/20 0.41
HSD17B3 P37058 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HRH3 Q9Y5N1 1/20 0.35
BRD4 O60885 1/20 0.34
ATAD2 Q6PL18 1/20 0.34
BAZ2B Q9UIF8 1/20 0.34
HSD17B10 Q99714 3/20 0.34
ALOX15 P16050 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798204 0.81 AKR1C3 (0.45) GABRA1GABRG2GABRB3MAPTKDM4E
SCHEMBL27593301 0.81 NR1H2 (0.50) NR1H2GABRA1GABRG2GABRB3MAPT
SCHEMBL218643 0.78 NR1H2 (0.48) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL1950813 0.77 HRH3 (0.48) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL30534578 0.77 HRH3 (0.48) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL8608562 0.76 NR1H2 (0.46) NR1H2GABRA1GABRG2GABRB3MAPT
SCHEMBL8798790 0.74 MAPT (0.46) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL24616867 0.71 HSD17B3 (0.42) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL2570232 0.71 HRH3 (0.49) NR1H2MAPTKDM4EALDH1A1LMNA
SCHEMBL397687 0.69 NR1H2 (0.66) NR1H2MAPTHSD17B3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790247-A1 TETRAHYDROISOQUINOLINE DERIVATIVE AND MEDICINAL PREPARATION CONTAINING THE SAME TERUMO KABUSHIKI KAISHA (JP) 1997-08-20 EP disclosed