SCHEMBL8608562

SCHEMBL8608562

CCOC(=O)CC(C)N1CCc2ccc(N)cc2C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.46
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HTT P42858 1/20 0.42
GABRA1 P14867 2/20 0.38
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
F10 P00742 7/20 0.38
PRSS1 P07477 7/20 0.38
PRSS2 P07478 7/20 0.38
PRSS3 P35030 7/20 0.38
F2 P00734 6/20 0.38
PLG P00747 6/20 0.38
HSD17B10 Q99714 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
POLB P06746 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8798709 0.82 DPP7 (0.48) KDM4EALDH1A1HTTGAAMAPT
SCHEMBL3910177 0.78 NR1H2 (0.49) NR1H2KDM4EALDH1A1HSD17B10MAPT
SCHEMBL38657715 0.78 TNF (0.41) NR1H2TMEM97SIGMAR1TNF
SCHEMBL8605349 0.76 TMEM97 (0.49) NR1H2KDM4EALDH1A1HTTGAA
SCHEMBL8798786 0.76 NR1H2 (0.49) NR1H2KDM4EALDH1A1GABRA1GABRG2
SCHEMBL27593301 0.74 NR1H2 (0.50) NR1H2KDM4EALDH1A1GABRA1GABRG2
SCHEMBL218643 0.74 NR1H2 (0.48) NR1H2KDM4EALDH1A1MAPTHTR1A
SCHEMBL30534578 0.74 HRH3 (0.48) NR1H2KDM4EALDH1A1GAAMAPT
SCHEMBL1950813 0.74 HRH3 (0.48) NR1H2KDM4EALDH1A1GAAMAPT
SCHEMBL1294235 0.73 NR1H2 (0.58) NR1H2KDM4EALDH1A1HTTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5789595-A ANTICOAGULANTS TERUMO KABUSHIKI KAISHA (JP) 1998-08-04 US disclosed
CN-1167485-A Tetrahydroisoquinoline derivative and medicinal preparation containing the same TERUMO CORP (JP) 1997-12-10 CN disclosed
EP-0790247-A1 TETRAHYDROISOQUINOLINE DERIVATIVE AND MEDICINAL PREPARATION CONTAINING THE SAME TERUMO KABUSHIKI KAISHA (JP) 1997-08-20 EP disclosed