SCHEMBL8799149

SCHEMBL8799149

Cc1cccc(Nc2cc(N[C@H]3CC[C@H](N(C)C)CC3)ncn2)c1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 13/20 0.50
EGFR P00533 5/20 0.50
TNNI3K Q59H18 3/20 0.48
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8799084 1.00 IRAK4 (0.50) IRAK4EGFRTNNI3KCYP1A2CYP3A4
SCHEMBL8798647 0.85 EGFR (0.55) IRAK4EGFRTNNI3K
SCHEMBL8798643 0.85 EGFR (0.55) IRAK4EGFRTNNI3K
SCHEMBL27318006 0.84 IRAK4 (0.42) IRAK4EGFRCYP1A2CYP3A4CYP2D6
SCHEMBL8801487 0.83 EGFR (0.50) EGFRTNNI3K
SCHEMBL8798907 0.83 EGFR (0.52) IRAK4EGFRTNNI3KCYP1A2CYP3A4
SCHEMBL8798928 0.82 EGFR (0.52) IRAK4EGFRTNNI3K
SCHEMBL8804869 0.82 EGFR (0.52) IRAK4EGFRTNNI3K
SCHEMBL8798922 0.82 EGFR (0.52) IRAK4EGFRTNNI3K
SCHEMBL8798960 0.82 EGFR (0.54) EGFRTNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed