SCHEMBL8799669

SCHEMBL8799669

COc1ccc2c(c1)N(C)C(Cl)=NS2(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
HTT P42858 2/20 0.42
GRIA2 P42262 2/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 1/20 0.35
NPC1 O15118 1/20 0.35
TDP1 Q9NUW8 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ELANE P08246 1/20 0.33
PTGES O14684 1/20 0.33
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10692092 0.72 NPC1 (0.43) CYP1A2CYP2C9CYP2C19HTTKDM4E
SCHEMBL18740669 0.69 PTGES (0.43) CYP1A2CYP2C9CYP2C19HTTKDM4E
SCHEMBL10571061 0.68 HTT (0.49) CYP1A2CYP2C9CYP2C19HTTMAPT
SCHEMBL10574320 0.67 TP53 (0.49) CYP1A2CYP2C9CYP2C19HTTKDM4E
SCHEMBL10572698 0.67 HTT (0.46) CYP1A2CYP2C9CYP2C19HTTMAPT
SCHEMBL10574780 0.67 CA12 (0.43) CYP1A2CYP2C9CYP2C19HTTKDM4E
SCHEMBL10572162 0.66 MAPT (0.46) CYP1A2CYP2C9CYP2C19HTTMAPT
SCHEMBL30808062 0.65 MEN1 (0.48) CYP1A2CYP2C9CYP2C19HTTHSD17B10
SCHEMBL26767749 0.65 CYP1A2 (0.62) CYP1A2CYP2C9CYP2C19HTTGRIA2
SCHEMBL10572752 0.64 HTT (0.51) CYP1A2CYP2C9CYP2C19HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641789-B1 BENZOTHIADIAZINE DERIVATIVE TAIHO PHARMACEUTICAL CO LTD (JP) 1997-12-03 EP disclosed
US-5401739-A Benzothiadiazine derivatives TAIHO PHARMACEUTICAL CO. LTD. (JP) 1995-03-28 US disclosed
EP-0641789-A1 BENZOTHIADIAZINE DERIVATIVE TAIHO PHARMACEUTICAL COMPANY LIMITED (JP) 1995-03-08 EP disclosed