SCHEMBL8799864

SCHEMBL8799864

CSc1cc(Nc2cccc(C)c2)ncn1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.57
TNNI3K Q59H18 5/20 0.54
NPSR1 Q6W5P4 1/20 0.46
HTT P42858 2/20 0.46
HIF1A Q16665 1/20 0.46
THRB P10828 1/20 0.46
RAB9A P51151 3/20 0.44
MAPK1 P28482 2/20 0.44
ERBB2 P04626 1/20 0.44
ABL1 P00519 1/20 0.44
ABL2 P42684 1/20 0.44
TSHR P16473 1/20 0.44
GFER P55789 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387302 0.85 EGFR (0.72) EGFRTNNI3KNPSR1HTTHIF1A
SCHEMBL8798667 0.83 EGFR (0.61) EGFRTNNI3KNPSR1HTTHIF1A
SCHEMBL2782010 0.80 EGFR (0.65) EGFRTNNI3KNPSR1HTTHIF1A
SCHEMBL2279629 0.78 EGFR (0.59) EGFRTNNI3KNPSR1HTTHIF1A
SCHEMBL7771269 0.77 EGFR (0.66) EGFRTNNI3KNPSR1HTTRAB9A
SCHEMBL8798959 0.77 EGFR (0.58) EGFRTNNI3KNPSR1HTTHIF1A
SCHEMBL690632 0.77 EGFR (0.62) EGFRTNNI3KHTTHIF1ARAB9A
SCHEMBL7777342 0.76 EGFR (0.64) EGFRTNNI3KNPSR1HTTHIF1A
SCHEMBL8798355 0.76 EGFR (0.60) EGFRTNNI3KNPSR1HTTHIF1A
SCHEMBL15197936 0.75 EGFR (0.56) EGFRTNNI3KNPSR1HTTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed