SCHEMBL8800657

SCHEMBL8800657

Nc1c(Cl)cc(Cl)cc1Nc1ncnc2cnc(N[C@H]3CC[C@H](O)CC3)nc12

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRAF P15056 7/20 0.56
EGFR P00533 1/20 0.50
ERBB2 P04626 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
MAPK3 P27361 2/20 0.42
ADORA1 P30542 2/20 0.41
ADORA2A P29274 1/20 0.39
CDK7 P50613 1/20 0.39
CDK9 P50750 1/20 0.39
MAPK14 Q16539 1/20 0.38
MAPK8 P45983 2/20 0.38
MAPK9 P45984 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993881 0.88 EGFR (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL6993890 0.88 EGFR (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL6996623 0.86 BRAF (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL6996614 0.86 BRAF (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL6999541 0.84 EGFR (0.52) BRAFEGFRERBB2HPGDHTT
SCHEMBL6999546 0.84 EGFR (0.52) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315973 0.81 EGFR (0.57) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315965 0.81 EGFR (0.57) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315344 0.80 EGFR (0.64) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315348 0.80 EGFR (0.64) BRAFEGFRERBB2HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed