SCHEMBL8800992

SCHEMBL8800992

O=C(O)Oc1cn(-c2cccc(Cn3cncn3)c2)c2nc(N3CCN(c4ccccc4)CC3)c(F)cc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.37
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
CYP2C9 P11712 1/20 0.36
ATP6V1B2 P21281 1/20 0.36
TBXA2R P21731 1/20 0.36
EDNRA P25101 1/20 0.36
TARBP2 Q15633 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
EPHA2 P29317 1/20 0.34
FLT4 P35916 1/20 0.34
GSK3B P49841 1/20 0.34
RARB P10826 1/20 0.34
TBXAS1 P24557 1/20 0.34
SLC6A3 Q01959 1/20 0.34
FAAH O00519 1/20 0.34
MGLL Q99685 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8800505 0.93 LMNA (0.37) CYP19A1KMT2ALMNACYP2C9ATP6V1B2
SCHEMBL8800987 0.92 KMT2A (0.45) CYP19A1KMT2ALMNACYP2C9ATP6V1B2
SCHEMBL8801716 0.91 LMNA (0.37) CYP19A1KMT2ALMNACYP2C9ATP6V1B2
SCHEMBL8802048 0.85 LMNA (0.42) CYP19A1KMT2ALMNAHDAC1HDAC6
SCHEMBL8801785 0.84 LMNA (0.37) KMT2ALMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8800501 0.84 LMNA (0.44) KMT2ALMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL8801651 0.79 CYP19A1 (0.37) CYP19A1KMT2ALMNAHDAC1HDAC6
SCHEMBL8803110 0.79 LMNA (0.37) CYP19A1KMT2ALMNACYP2C9ATP6V1B2
SCHEMBL8801047 0.78 LMNA (0.46) KMT2ALMNAKDM4EMEN1ALDH1A1
SCHEMBL9058127 0.78 HDAC1 (0.37) CYP19A1HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612731-B1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1997-08-20 EP disclosed
EP-0612731-A1 Novel guinolone and naphthyridone derivatives BAYER AG (DE) 1994-08-31 EP disclosed