SCHEMBL8801424

SCHEMBL8801424

COC(=O)Oc1cccc2[nH]ccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 2/20 0.50
HTR1A P08908 7/20 0.49
CYP1A2 P05177 2/20 0.49
CYP3A4 P08684 2/20 0.49
LMNA P02545 2/20 0.49
ADRB2 P07550 2/20 0.49
ADRB1 P08588 2/20 0.49
ADRB3 P13945 2/20 0.49
KDM4E B2RXH2 2/20 0.49
USP2 O75604 1/20 0.49
CYP2D6 P10635 1/20 0.49
THRB P10828 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
TP53 P04637 1/20 0.49
GLA P06280 1/20 0.49
ALOX15 P16050 1/20 0.49
NFKB1 P19838 1/20 0.49
DRD4 P21917 1/20 0.49
HTR2C P28335 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29511854 0.83 SLC22A6 (0.63) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL594038 0.83 SLC22A6 (0.63) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL12543813 0.83 HTR1A (0.43) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL30733595 0.83 HTR1A (0.50) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL7495860 0.83 BCHE (0.60) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL29938170 0.83 BCHE (0.60) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL2312464 0.81 RHEB (0.49) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL29966634 0.81 HTR1A (0.52) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL9871925 0.80 RHEB (0.51) HTR1BHTR1ACYP1A2CYP3A4LMNA
SCHEMBL8583050 0.79 SLC22A6 (0.46) HTR1BHTR1ACYP1A2CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525584-B1 6-Oxo-azepinoindole derivatives, process and intermediates for their preparation and medicaments containing them SOLVAY PHARM GMBH (DE) 1997-12-10 EP disclosed
EP-0525584-A1 6-Oxo-azepinoindole derivatives, process and intermediates for their preparation and medicaments containing them Kali-Chemie Pharma GmbH (DE) 1993-02-03 EP disclosed