SCHEMBL8801548

SCHEMBL8801548

Cc1ccc(Cl)c2[nH]c3c(c12)CCNC3

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.44
NISCH Q9Y2I1 3/20 0.42
KDM4E B2RXH2 1/20 0.40
HTR5A P47898 1/20 0.40
NR2E1 Q9Y466 1/20 0.40
HTT P42858 1/20 0.39
PTK2B Q14289 1/20 0.39
PNMT P11086 5/20 0.38
ADRA2A P08913 3/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
CLCN2 P51788 1/20 0.38
HTR7 P34969 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
THRB P10828 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14581535 0.88 TAAR1 (0.55) TAAR1HTTPTK2BPNMTADRA2A
Hydrochloric Acid SCHEMBL4792618 0.87 TAAR1 (0.57) TAAR1HTTPTK2BPNMTADRA2A
SCHEMBL6823728 0.81 ADRA2A (0.38) TAAR1KDM4EHTTPTK2BADRA2A
SCHEMBL4793578 0.79 TAAR1 (0.51) TAAR1NISCHHTTPTK2BPNMT
Hydrochloric Acid SCHEMBL4792338 0.78 TAAR1 (0.54) TAAR1NISCHHTTPTK2BPNMT
SCHEMBL14581525 0.78 TAAR1 (0.45) TAAR1NISCHKDM4EHTR5ANR2E1
SCHEMBL31020934 0.78 TAAR1 (0.45) TAAR1NISCHKDM4EHTR5ANR2E1
Hydrochloric Acid SCHEMBL4791753 0.76 TAAR1 (0.48) TAAR1NISCHKDM4EHTR5ANR2E1
SCHEMBL8814257 0.76 NISCH (0.52) TAAR1NISCHKDM4EHTR5ANR2E1
SCHEMBL8802563 0.76 NISCH (0.56) TAAR1NISCHKDM4EHTR5ANR2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751770-A4 8-SUBSTITUTED TETRAHYDRO-BETA-CARBOLINES LILLY CO ELI (US) 1997-06-11 EP disclosed
EP-0751770-A1 8-SUBSTITUTED TETRAHYDRO-BETA-CARBOLINES ELI LILLY AND COMPANY (US) 1997-01-08 EP disclosed
WO-1995024191-A1 8-SUBSTITUTED TETRAHYDRO-BETA-CARBOLINES ELI LILLY AND COMPANY (US) 1995-09-14 WO disclosed