SCHEMBL8801593

SCHEMBL8801593

CC(C)(C)OC(=O)c1n[nH]c2nc(N3CCNCC3)ccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HRH4 Q9H3N8 4/20 0.41
ACACB O00763 1/20 0.40
ACACA Q13085 1/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
HRH3 Q9Y5N1 2/20 0.38
PARP1 P09874 2/20 0.38
CYP3A4 P08684 2/20 0.37
HSD17B10 Q99714 2/20 0.37
AURKA O14965 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
USP2 O75604 1/20 0.36
HTR3B O95264 1/20 0.36
CYP1A2 P05177 1/20 0.36
ADRB1 P08588 1/20 0.36
HTR1A P08908 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801559 0.89 ALDH1A1 (0.39) KDM4EMEN1KMT2AHRH4ALDH1A1
SCHEMBL25343179 0.86 PTGER4 (0.40) HRH4ACACBALDH1A1LMNAMAPK1
SCHEMBL30526303 0.86 PTGER4 (0.40) HRH4ACACBALDH1A1LMNAMAPK1
SCHEMBL491961 0.83 TRPV1 (0.41) ALDH1A1LMNAAURKAFGFR1
SCHEMBL8801585 0.82 KDM4E (0.45) KDM4EMEN1KMT2AHRH4ALDH1A1
SCHEMBL8801084 0.81 IRAK4 (0.45) KDM4EALDH1A1HRH3PARP1CYP3A4
Hydrochloric Acid SCHEMBL8801958 0.79 IRAK4 (0.43) KDM4EMEN1KMT2AALDH1A1HRH3
SCHEMBL8800895 0.76 KDM4E (0.47) KDM4EMEN1KMT2AHRH4ALDH1A1
SCHEMBL30526295 0.75 ALDH1A1 (0.45) KDM4EMEN1KMT2AALDH1A1LMNA
SCHEMBL492450 0.75 ALDH1A1 (0.45) KDM4EMEN1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5300498-A Treating depression, obsessive compulsive disorder HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-04-05 US claimed
EP-0627432-B1 6-Piperazinyl-1H-pyrazolo [3,4-b]pyridine-3-carboxylic Acids, Esters, Amides and related compounds, a process for their preparation and their use as medicaments HOECHST MARION ROUSSEL INC (US) 1997-09-03 EP disclosed
EP-0627432-A1 6-Piperazinyl-1H-pyrazolo [3,4-b]pyridine-3-carboxylic Acids, Esters, Amides andrelated compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-12-07 EP disclosed
US-5300498-A Treating depression, obsessive compulsive disorder HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-04-05 US disclosed