SCHEMBL8802190

SCHEMBL8802190

C#Cc1c(N2CC3NCCOC3C2)c(F)cc2c(=O)c(OC(=O)O)cn(C3CC3)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
KDM4E B2RXH2 4/20 0.45
HPGD P15428 4/20 0.45
HSD17B10 Q99714 3/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KCNH2 Q12809 6/20 0.41
POLB P06746 2/20 0.41
OPRM1 P35372 2/20 0.41
PRKD3 O94806 1/20 0.41
ALOX15 P16050 1/20 0.41
CLK2 P49760 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
OPRD1 P41143 1/20 0.36
SSTR2 P30874 3/20 0.35
LMNA P02545 2/20 0.34
TOP2A P11388 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610667 0.92 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7608350 0.92 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7608326 0.92 ALDH1A1 (0.45) ALDH1A1KDM4EHPGDHSD17B10MEN1
Hydrochloric Acid SCHEMBL7608719 0.92 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10MEN1
Hydrochloric Acid SCHEMBL7615492 0.92 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL9182746 0.90 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL8803776 0.90 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL8330927 0.90 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL6217934 0.90 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHSD17B10MEN1
Hydrochloric Acid SCHEMBL8329739 0.89 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0523512-B1 8-vinyl- and 8-ethinyl-quinolone carboxylic acids BAYER AG (DE) 1997-01-15 EP claimed
EP-0523512-A1 8-vinyl- and 8-ethinyl-quinolone carboxylic acids BAYER AG (DE) 1993-01-20 EP claimed
EP-0523512-B1 8-vinyl- and 8-ethinyl-quinolone carboxylic acids BAYER AG (DE) 1997-01-15 EP disclosed
EP-0523512-A1 8-vinyl- and 8-ethinyl-quinolone carboxylic acids BAYER AG (DE) 1993-01-20 EP disclosed