SCHEMBL8804145

SCHEMBL8804145

CN1CC2CC(NC(=O)Nc3ccccc3C=Cc3cc(C(C)(C)C)c(O)c(C(C)(C)C)c3)CC(C1)N2C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.40
MAOB P27338 3/20 0.40
PTGS1 P23219 4/20 0.36
PTGS2 P35354 4/20 0.36
ALOX5 P09917 2/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
SNCA P37840 1/20 0.34
P2RY1 P47900 1/20 0.34
ALPL P05186 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8803421 0.82 KMT2A (0.53) MAOAMAOBP2RY1
SCHEMBL8803427 0.82 KMT2A (0.53) MAOAMAOBP2RY1
SCHEMBL8804441 0.80 CYP2D6 (0.42) MAOAMAOBCYP2D6CYP2C19ACHE
SCHEMBL8803896 0.78 P2RY1 (0.52) MAOAMAOBPTGS1PTGS2ALOX5
SCHEMBL8803557 0.76 KDM4E (0.48) MAOAMAOBPTGS1PTGS2ALOX5
SCHEMBL8803559 0.76 KDM4E (0.48) MAOAMAOBPTGS1PTGS2ALOX5
SCHEMBL8803889 0.74 EPHX2 (0.54)
SCHEMBL8803890 0.74 EPHX2 (0.54)
Hydrochloric Acid SCHEMBL8946231 0.74 F10 (0.42)
SCHEMBL8805752 0.72 CYP2D6 (0.48) MAOAMAOBCYP2D6CYP2C19ALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625507-B1 Urea derivatives and their use as acat inhibitors NISSHIN FLOUR MILLING CO (JP) 1997-07-23 EP disclosed
US-5621010-A ANTIHYPERCHOLESTEROLEMIA AND ANTIATHEROSCLEROSIS NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-04-15 US disclosed
EP-0625507-A2 Urea derivatives and their use as acat inhibitors NISSHIN FLOUR MILLING CO., LTD. (JP) 1994-11-23 EP disclosed