SCHEMBL880548

SCHEMBL880548

CC(O)C(=O)C1(O)CCNCC1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
KDM4E B2RXH2 1/20 0.35
KMT2A Q03164 1/20 0.35
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6914016 0.86 CYP1A2 (0.38) CYP1A2KDM4EKMT2A
SCHEMBL6915421 0.74 CYP1A2 (0.33) CYP1A2KDM4EKMT2A
SCHEMBL1282200 0.74 KDM4E (0.37) CYP1A2KDM4EKMT2A
Hydrochloric Acid SCHEMBL5750787 0.72 KDM4E (0.35) KDM4EKMT2A
SCHEMBL7286601 0.72 KDM4E (0.40) CYP1A2KDM4EKMT2A
SCHEMBL888643 0.68
SCHEMBL61405 0.67 KDM4E (0.50) KDM4EKMT2A
SCHEMBL854175 0.67 KDM4E (0.41) CYP1A2KDM4EKMT2A
SCHEMBL19035187 0.67 CYP1A2 (0.37) CYP1A2KDM4EKMT2A
Piperazine SCHEMBL7553577 0.66 TP53 (0.65) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2433937-A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof Purdue Pharma LP (US) 2012-03-28 EP disclosed
EP-2433935-A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof Purdue Pharma LP (US) 2012-03-28 EP disclosed
EP-2433936-A1 Substituted-quinoxaline-type-piperidine compounds and the uses thereof Purdue Pharma LP (US) 2012-03-28 EP disclosed
WO-2009027820-A2 SUBSTITUTED-QUINOXALINE-TYPE-PIPERIDINE COMPOUNDS AND THE USES THEREOF PURDUE PHARMA L.P. (DE) 2009-03-05 WO disclosed