SCHEMBL1282200

SCHEMBL1282200

O=C(O)C1(O)CCNCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 1/20 0.37
OPRM1 P35372 2/20 0.36
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
TSHR P16473 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRE P78334 1/20 0.35
PMP22 Q01453 1/20 0.35
GABRA6 Q16445 1/20 0.35
GABRG1 Q8N1C3 1/20 0.35
GABRG3 Q99928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5750787 0.97 KDM4E (0.35) KDM4EKMT2AOPRM1GABRPGABRD
SCHEMBL1855601 0.84
Hydrochloric Acid SCHEMBL11546148 0.82 HTR2A (0.34)
SCHEMBL28736616 0.82 KDM4E (0.35) KDM4EKMT2AOPRM1
Toluene SCHEMBL27914297 0.80 OPRM1 (0.46) KMT2AOPRM1GABRDGABRA1TSHR
SCHEMBL153693 0.78
SCHEMBL61405 0.76 KDM4E (0.50) KDM4EKMT2AOPRM1DRD2
SCHEMBL7286601 0.76 KDM4E (0.40) KDM4EKMT2AOPRM1GABRDGABRA1
SCHEMBL6757053 0.76
SCHEMBL825722 0.74 KDM4E (0.38) KDM4EKMT2AOPRM1GABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 146 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114349922-A Flexible dual-curing resin composition and preparation method of forming body thereof 浙江华峰新材料有限公司 2022-04-15 CN claimed
CN-109863146-A Aryl-linking compound as immunomodulator 百时美施贵宝公司 2019-06-07 CN claimed
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GENZYME CORPORATION (US) 2025-01-23 US disclosed
US-12180226-B2 Spirotricycle RIPK1 inhibitors and methods of uses thereof MERCK SHARP & DOHME LLC (US) 2024-12-31 US disclosed
EP-4423096-A1 SPIROTRICYCLE RIPK1 INHIBITORS AND METHODS OF USES THEREOF Merck Sharp & Dohme LLC (US) 2024-09-04 EP disclosed
US-20240277706-A1 METHODS AND COMPOSTITIONS FOR TARGETING PD-L1 ALIGOS THERAPEUTICS, INC. 2024-08-22 US disclosed
US-12060349-B2 Glucosylceramide synthase inhibitors GENZYME CORPORATION (US) 2024-08-13 US disclosed
CN-118488957-A Spirotricyclic RIPK1 inhibitors and methods of use thereof 默沙东有限责任公司 2024-08-13 CN disclosed
US-20230348427-A1 COMPOUND FOR ANDROGEN RECEPTOR DEGRADATION, AND PHARMACEUTICAL USE THEREOF UBIX THERAPEUTICS, INC. (KR) 2023-11-02 US disclosed
EP-3998260-B1 SGC STIMULATORS CYCLERION THERAPEUTICS INC (US) 2023-11-01 EP disclosed
EP-4240736-A1 PPAR GAMMA MODULATORS AND METHODS OF USE Eisai R&D Management Co., Ltd. (JP) 2023-09-13 EP disclosed
US-6576627-B1 Such as 7-amino-2-((2-methyl-1-(3-phenylpropanoylamino)-propyl)hydroxyphosphinoyl) -methylheptanoic acid; thrombotic disease MEIJI SEIKA KAISHA LTD. (JP) 2003-06-10 US disclosed
EP-1152004-B1 Phosphonic acid derivatives having carboxypeptidase B inhibitory action MEIJI SEIKA KAISHA (JP) 2003-05-07 EP disclosed
WO-2003010138-A2 PIPERIDINE DERIVATIVES AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2003-02-06 WO disclosed
CN-1373766-A Phosphonic acid derivatives having carboxypeptidase B inhibitory activity MEIJI SEIKA KAISHA (JP) 2002-10-09 CN disclosed
EP-1174434-A1 Phosphonic acid derivative having inhibitory activity against carboxypeptidase B MEIJI SEIKA KAISHA LTD. (JP) 2002-01-23 EP disclosed
EP-1152004-A1 PHOSPHONIC ACID DERIVATIVES HAVING CARBOXYPEPTIDASE B INHIBITORY ACTIVITY MEIJI SEIKA KAISHA LTD. (JP) 2001-11-07 EP disclosed
CN-1052231-C Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2000-05-10 CN disclosed
CN-1097421-A Adhesion receptor antagonists MERCK PATENT GMBH (DE) 1995-01-18 CN disclosed
US-4247694-A PHOTOSTABILIZERS FOR POLYMERS CIBA-GEIGY CORPORATION (US) 1981-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240277706-A1 METHODS AND COMPOSTITIONS FOR TARGETING PD-L1 CD274, PDCD1, PDCD1LG2 KDM4E 2919/4885KMT2A 2875/4885OPRM1 2759/4885
US-20230348427-A1 COMPOUND FOR ANDROGEN RECEPTOR DEGRADATION, AND PHARMACEUTICAL USE THEREOF AR, NR5A1, SHBG KDM4E 2263/4885KMT2A 2131/4885OPRM1 984/4885
US-12060349-B2 Glucosylceramide synthase inhibitors GBA1, GBA2, GALC KDM4E 4213/4885KMT2A 2942/4885OPRM1 4766/4885
US-20250026749-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS GBA1, GBA2, GAA KDM4E 4241/4885KMT2A 2721/4885OPRM1 4772/4885
US-12180226-B2 Spirotricycle RIPK1 inhibitors and methods of uses thereof RIPK1, RIPK3, RIPK4 KDM4E 3571/4885KMT2A 3659/4885OPRM1 4667/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.