SCHEMBL8806366

SCHEMBL8806366

O=C(O)c1c(O)c2ccc([N+](=O)[O-])cc2[nH]c1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.58
GRIA1 P42261 1/20 0.53
GRIA2 P42262 1/20 0.53
GRIA3 P42263 1/20 0.53
GRIA4 P48058 1/20 0.53
FASN P49327 1/20 0.51
DAO P14920 1/20 0.50
GRIN2D O15399 1/20 0.49
GRIN3B O60391 1/20 0.49
GRIN1 Q05586 1/20 0.49
GRIN2A Q12879 1/20 0.49
GRIN2B Q13224 1/20 0.49
GRIN2C Q14957 1/20 0.49
GRIN3A Q8TCU5 1/20 0.49
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
PKM P14618 1/20 0.47
NPY1R P25929 1/20 0.47
NPY2R P49146 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10651016 0.87 PARP1 (0.53) PARP1GRIA1GRIA2GRIA3GRIA4
SCHEMBL8136947 0.85 PARP1 (0.55) PARP1GRIA1GRIA2GRIA3GRIA4
SCHEMBL8000855 0.84 PARP1 (0.67) PARP1GRIA1GRIA2GRIA3GRIA4
SCHEMBL5309020 0.83 SERPINE1 (0.50) PARP1GRIA1GRIA2GRIA3GRIA4
SCHEMBL5334737 0.81 KDM5A (0.58) PARP1GRIA1GRIA2GRIA3GRIA4
SCHEMBL8785378 0.78 FASN (0.81) PARP1FASNDAOGRIN2DGRIN3B
SCHEMBL10650769 0.78 PARP1 (0.46) PARP1GRIA1GRIA2GRIA3GRIA4
SCHEMBL11107841 0.78 KDM4E (0.50) PARP1FASNMEN1ALDH1A1POLB
SCHEMBL8000790 0.77 PARP1 (0.57) PARP1GRIA1GRIA2GRIA3GRIA4
SCHEMBL8139112 0.77 MEN1 (0.70) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760819-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-03-12 EP disclosed
WO-1995032205-A1 TRICYCLIC DICARBONYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1995-11-30 WO disclosed