SCHEMBL8807100

SCHEMBL8807100

Cc1cc2ncnc(O)c2cc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.41
CSF1R P07333 2/20 0.41
KDM4E B2RXH2 2/20 0.40
MAPT P10636 2/20 0.40
IRAK4 Q9NWZ3 2/20 0.40
RET P07949 8/20 0.34
KDR P35968 7/20 0.34
KIF5B P33176 6/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
RAD52 P43351 1/20 0.33
RAB9A P51151 1/20 0.33
QRFPR Q96P65 1/20 0.33
FGFR1 P11362 1/20 0.33
FLT1 P17948 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
ALDH1A1 P00352 1/20 0.32
NQO2 P16083 1/20 0.32
GAK O14976 1/20 0.31
RIPK2 O43353 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20355005 0.84 JAK3 (0.35) EGFRCSF1RKDM4EMAPTIRAK4
SCHEMBL25552038 0.84 EGFR (0.40) EGFRCSF1RMAPTIRAK4RET
SCHEMBL16016669 0.81 RET (0.47) EGFRCSF1RIRAK4RETKDR
SCHEMBL25873553 0.80 GABRP (0.41) KDM4ESMN1; SMN2LMNAALDH1A1
SCHEMBL25873554 0.80 SMN1; SMN2 (0.36) KDM4EMAPTKDRSMN1; SMN2HTT
SCHEMBL14579634 0.77 GAA (0.42) EGFRMAPTALDH1A1
SCHEMBL12703881 0.77 EGFR (0.44) EGFRCSF1RKDM4EMAPTIRAK4
SCHEMBL18013039 0.77 EGFR (0.42) EGFRIRAK4RETKDRKIF5B
SCHEMBL15890160 0.76 GAK (0.39) GAKRIPK2
SCHEMBL1012225 0.75 HTT (0.50) KDM4EMAPTIRAK4SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed