SCHEMBL8807306

SCHEMBL8807306

NC(=O)OC1(c2ccccc2)CCN(CCC2(c3ccc(Cl)c(Cl)c3)CC(=O)N(Cc3ccccc3)C2)CC1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.63
CCR5 P51681 2/20 0.61
TACR2 P21452 4/20 0.56
TACR3 P29371 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8351334 0.87 TACR1 (0.66) TACR1CCR5TACR2TACR3
SCHEMBL8347309 0.85 TACR1 (0.68) TACR1CCR5TACR2TACR3
SCHEMBL8808304 0.81 TACR2 (0.77) TACR1TACR2TACR3
SCHEMBL7770397 0.78 TACR1 (0.75) TACR1CCR5TACR2TACR3
SCHEMBL7764193 0.78 TACR1 (0.72) TACR1CCR5TACR2TACR3
SCHEMBL7306896 0.77 TACR1 (1.00) TACR1CCR5TACR2TACR3
Hydrochloric Acid SCHEMBL8483004 0.77 TACR1 (0.74) TACR1CCR5TACR2TACR3
Hydrochloric Acid SCHEMBL8480218 0.77 TACR1 (0.71) TACR1CCR5TACR2TACR3
SCHEMBL8355624 0.77 TACR1 (0.52) TACR1CCR5TACR2TACR3
SCHEMBL7956540 0.77 CCR5 (0.58) TACR1CCR5TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696280-B1 SUBSTITUTED PYRROLIDIN-3-YL-ALKYL-PIPERIDINES USEFUL AS TACHYKININ ANTAGONISTS MERRELL PHARMA INC (US) 1997-09-24 EP claimed