SCHEMBL8809131

SCHEMBL8809131

N=C(N)c1ccc(CNC(=O)[C@@H]2CCCN2)cc1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.64
HTR2B P41595 3/20 0.64
F2 P00734 9/20 0.60
KDM4E B2RXH2 1/20 0.57
HDAC1 Q13547 3/20 0.55
HDAC3 O15379 2/20 0.52
HDAC2 Q92769 1/20 0.52
MASP2 O00187 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5900833 0.99 HTR2C (0.62) HTR2CHTR2BF2KDM4EHDAC1
Hydrochloric Acid SCHEMBL5900838 0.99 HTR2C (0.62) HTR2CHTR2BF2KDM4EHDAC1
SCHEMBL6606024 0.93 F2 (0.61) HTR2CHTR2BF2MASP2
SCHEMBL23840789 0.85 F2 (0.72) F2MASP2
SCHEMBL23793372 0.85 F2 (0.59) HTR2CHTR2BF2MASP2
SCHEMBL17268026 0.84 HTR2C (0.70) HTR2CHTR2BKDM4EHDAC1HDAC3
SCHEMBL8305420 0.83 PRCP (0.47) HTR2CHTR2BF2KDM4EHDAC1
SCHEMBL24653087 0.81 HTR2C (0.70) HTR2CHTR2BKDM4EHDAC1HDAC3
SCHEMBL24648976 0.81 HTR2C (0.70) HTR2CHTR2BKDM4EHDAC1HDAC3
SCHEMBL21206860 0.81 HTR2C (0.70) HTR2CHTR2BKDM4EHDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355674-B1 OLIGO ALKYLENE GLYCOL OR POLYALKYLENE GLYCOL-COUPLED THROMBIN INHIBITORS JENAFFIN GMBH (DE) 2010-10-27 EP disclosed
WO-1996025426-A9 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS 1997-06-12 WO disclosed