SCHEMBL8809376

SCHEMBL8809376

Oc1ncnc2cc(C(F)(F)F)ccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.49
KDM4E B2RXH2 1/20 0.46
EGFR P00533 8/20 0.43
ADRB2 P07550 1/20 0.41
NCF1 P14598 1/20 0.41
PKM P14618 1/20 0.40
ABCG2 Q9UNQ0 2/20 0.39
MAOB P27338 1/20 0.39
SCN9A Q15858 1/20 0.39
DYRK3 O43781 2/20 0.39
GSK3A P49840 2/20 0.39
GSK3B P49841 2/20 0.39
DYRK1A Q13627 2/20 0.39
CLK4 Q9HAZ1 2/20 0.39
STK17A Q9UEE5 2/20 0.39
PLK4 O00444 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
CHEK2 O96017 1/20 0.39
FGFR1 P11362 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL686726 0.86 KDM4E (0.46) KDM4EEGFRABCG2KDRTSHR
SCHEMBL26313476 0.79 PARP1 (0.49) PARP1KDM4EEGFRADRB2NCF1
SCHEMBL27461883 0.79 PARP1 (0.49) PARP1KDM4EEGFRADRB2NCF1
SCHEMBL26090047 0.79 PARP1 (0.49) PARP1KDM4EEGFRADRB2NCF1
SCHEMBL29416609 0.79 PARP1 (0.49) PARP1KDM4EEGFRADRB2NCF1
SCHEMBL857761 0.79 PARP1 (0.49) PARP1KDM4EEGFRADRB2NCF1
SCHEMBL28066432 0.77 EGFR (0.37) PARP1EGFRKDR
SCHEMBL1766094 0.76 CSF1R (0.42) KDM4EEGFRABCG2MAP4K4FGFR1
SCHEMBL31549968 0.76 CSF1R (0.42) KDM4EEGFRABCG2MAP4K4FGFR1
SCHEMBL2345433 0.75 ADRB2 (0.51) PARP1KDM4EADRB2NCF1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782570-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1997-07-09 EP disclosed
WO-1996009294-A1 SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE IN MEDICINE THE WELLCOME FOUNDATION LIMITED (GB) 1996-03-28 WO disclosed