SCHEMBL8809652

SCHEMBL8809652

NC(=O)c1cccc(-c2ccccc2)c1-c1ccsc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.57
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
HNF4A P41235 1/20 0.46
CYP2E1 P05181 1/20 0.46
CYP2A6 P11509 1/20 0.46
CYP2B6 P20813 1/20 0.46
IKBKB O14920 5/20 0.42
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PDK2 Q15119 1/20 0.40
CCNE2 O96020 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
CHUK O15111 1/20 0.40
IKBKE Q14164 1/20 0.40
PKMYT1 Q99640 1/20 0.40
CHEK1 O14757 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2025737 0.85 BCAT2 (0.71) BCAT2KEAP1NFE2L2HNF4AIKBKB
Hydrochloric Acid SCHEMBL27966297 0.84 BCAT2 (0.69) BCAT2KEAP1NFE2L2HNF4AIKBKB
SCHEMBL4481912 0.82 BCAT2 (0.61) BCAT2KEAP1NFE2L2CYP2E1CYP2A6
SCHEMBL8812799 0.82 GRM5 (0.47) BCAT2KEAP1NFE2L2IKBKBCCNE2
Hydrochloric Acid SCHEMBL27721971 0.81 BCAT2 (0.59) BCAT2KEAP1NFE2L2CYP2E1CYP2A6
Phosphoric Acid SCHEMBL3689008 0.80 BCAT2 (0.62) BCAT2KEAP1NFE2L2HNF4AIKBKB
SCHEMBL28309328 0.78 BCAT2 (0.43) BCAT2KEAP1NFE2L2CYP2E1CYP2A6
SCHEMBL27510657 0.77 CYP2A6 (0.59) HNF4ACYP2E1CYP2A6CYP2B6PDK2
SCHEMBL30370009 0.76 BCAT2 (0.57) BCAT2KEAP1NFE2L2HNF4AIKBKB
Thiophene SCHEMBL28606237 0.76 BCAT2 (0.79) BCAT2KEAP1NFE2L2HNF4AIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804420-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-11-05 EP disclosed