SCHEMBL8810459

SCHEMBL8810459

CCOC(=O)CC[C@@H]1C(=O)N(c2ccc(OC)cc2)[C@@H]1C(=O)OC

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
KDM4E B2RXH2 2/20 0.50
HPGD P15428 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.45
NPSR1 Q6W5P4 1/20 0.44
GAA P10253 2/20 0.41
POLB P06746 1/20 0.39
TP53 P04637 1/20 0.39
KLK7 P49862 1/20 0.39
TSHR P16473 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALOX15 P16050 1/20 0.39
P2RX3 P56373 4/20 0.39
SOAT1 P35610 1/20 0.39
CYP2C9 P11712 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8810449 1.00 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDSMN1; SMN2NPSR1
SCHEMBL8810455 1.00 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDSMN1; SMN2NPSR1
SCHEMBL5632939 0.85 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL7434157 0.83 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL7434354 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL17977269 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL8260150 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL7430439 0.76 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL7436135 0.76 ALDH1A1 (0.53) ALDH1A1KDM4EHPGDSMN1; SMN2GAA
SCHEMBL8812717 0.75 SOAT1 (0.44) ALDH1A1KDM4EHPGDNPSR1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997013750-A1 AZETIDINONES AND THEIR THERAPEUTIC USE AS CYTOKINE INHIBITORS CHIROSCIENCE LIMITED (GB) 1997-04-17 WO disclosed