SCHEMBL881069

SCHEMBL881069

Nn1nc2c(c1C(=O)O)CCc1cc(O)ccc1-2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.45
CYP2C9 P11712 5/20 0.41
CYP2C8 P10632 4/20 0.40
S1PR1 P21453 3/20 0.40
AKR1B1 P15121 2/20 0.39
MAOB P27338 2/20 0.37
MAOA P21397 1/20 0.37
PRKCI P41743 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALPL P05186 1/20 0.37
CLK1 P49759 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
HSP90AA1 P07900 1/20 0.37
PTAFR P25105 1/20 0.36
MIF P14174 2/20 0.36
ESR2 Q92731 1/20 0.35
SRD5A1 P18405 1/20 0.35
SRD5A2 P31213 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6792714 0.84 HCAR2 (0.55) HCAR2CYP2C9CYP2C8S1PR1AKR1B1
Hydrochloric Acid SCHEMBL1656581 0.79 HCAR2 (0.44) HCAR2CYP2C9CYP2C8S1PR1AKR1B1
SCHEMBL6791799 0.78 HCAR2 (0.43) HCAR2CYP2C9CYP2C8S1PR1AKR1B1
SCHEMBL6793335 0.78 HCAR2 (0.49) HCAR2CYP2C9CYP2C8S1PR1AKR1B1
SCHEMBL6792867 0.71 HCAR2 (0.56) HCAR2CYP2C9CYP2C8AKR1B1MAOB
SCHEMBL6786891 0.71 HCAR2 (0.48) HCAR2CYP2C9S1PR1KDM4EMEN1
SCHEMBL6795109 0.70 MEN1 (0.69) HCAR2CYP2C9CYP2C8S1PR1AKR1B1
SCHEMBL6793002 0.69 HCAR2 (0.41) HCAR2CYP2C9CYP2C8AKR1B1ESR2
SCHEMBL19128564 0.68 KDM4E (0.59) CYP2C9KDM4EMEN1ALPLCLK1
Bromide SCHEMBL6799686 0.68 HCAR2 (0.41) HCAR2CYP2C9CYP2C8AKR1B1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2433496-A1 Tissue non-specific alkaline phosphatase inhibitors and uses thereof for treating vascular calcification Burnham Institute for Medical Research (US) 2012-03-28 EP disclosed