SCHEMBL8818671

SCHEMBL8818671

COc1ncccc1-c1nc(-c2cccc(C)n2)nc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 9/20 0.49
MAPK14 Q16539 2/20 0.49
DHODH Q02127 1/20 0.45
MAPT P10636 5/20 0.45
NPSR1 Q6W5P4 2/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.42
LMNA P02545 1/20 0.42
RECQL P46063 1/20 0.42
POLB P06746 1/20 0.41
ABCB1 P08183 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
ELANE P08246 1/20 0.40
METAP1 P53582 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8816582 0.83 ADORA2A (0.58) TGFBR1MAPK14MAPTNPSR1ALDH1A1
SCHEMBL8818694 0.80 ADORA2A (0.48) TGFBR1MAPK14MAPTNPSR1ALDH1A1
SCHEMBL8818444 0.80 ADORA2A (0.56) TGFBR1MAPK14MAPTALDH1A1LMNA
SCHEMBL8815685 0.80 TGFBR1 (0.51) TGFBR1MAPK14ALDH1A1
SCHEMBL8818479 0.79 ADORA2A (0.47) TGFBR1MAPK14MAPTNPSR1ALDH1A1
SCHEMBL8818575 0.78 ADORA2A (0.43) TGFBR1MAPK14ALDH1A1
SCHEMBL22939929 0.78 CCR1 (0.48) TGFBR1L3MBTL1ELANE
SCHEMBL8818439 0.78 TGFBR1 (0.49) TGFBR1MAPK14MAPTL3MBTL1ABCB1
SCHEMBL8815690 0.78 TGFBR1 (0.49) TGFBR1MAPK14ALDH1A1
SCHEMBL8818447 0.78 ADORA2A (0.54) TGFBR1MAPK14MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012066122-A1 2 - (PYRIDIN- 2 -YL) -QUINAZOLINE DERIVATIVES AND THEIR USE AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-24 WO disclosed