SCHEMBL8823764

SCHEMBL8823764

COc1cccc2c1CCCO2

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.49
HTR1A P08908 2/20 0.42
DRD2 P14416 1/20 0.42
DRD1 P21728 1/20 0.42
HTR1B P28222 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
CTNNB1 P35222 2/20 0.40
WNT3A P56704 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8823797 0.85 BCHE (0.48) ACHEDRD2
Hydrochloric Acid SCHEMBL8823770 0.84 BCHE (0.47) ACHEDRD2
SCHEMBL16659183 0.81 HTR2C (0.37) ACHEHTR1AHTR1BHTR2AHTR2C
SCHEMBL27640856 0.79 MTNR1A (0.48) ACHE
SCHEMBL29054671 0.78 MTNR1A (0.41) ACHEHTR1ADRD2HTR1BHTR2A
SCHEMBL436160 0.77 MAP3K14 (0.46) ACHEHTR1AHTR1BHTR2AHTR2C
SCHEMBL6621347 0.77 MTNR1A (0.44)
SCHEMBL19756701 0.76 HTR2C (0.38) ACHEHTR1AHTR1BHTR2AHTR2C
SCHEMBL12239586 0.76 MTNR1A (0.43) ACHECTNNB1WNT3A
SCHEMBL21872018 0.75 MTNR1A (0.47) HTR1AHTR1BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240167066-A1 METHOD FOR PRODUCING DEMETHYLATED COMPOUND DAICEL CORPORATION (JP) 2024-05-23 US disclosed
WO-2022202961-A1 METHOD FOR PRODUCING DEMETHYLATED COMPOUND 株式会社ダイセル 2022-09-29 WO disclosed
US-5656657-A Chroman derivatives ASTRA AKTIEBOLAG (SE) 1997-08-12 US disclosed
US-5656658-A Method for the treatment of anxiety ASTRA AKTIEBOLAG (SE) 1997-08-12 US disclosed
US-5650524-A Process for preparing (R)-3-amino-5-methoxychroman ASTRA AKTIEBOLAG (SE) 1997-07-22 US disclosed
US-5646309-A Intermediates in the synthesis of chroman derivatives ASTRA AKTIEBOLAG (SE) 1997-07-08 US disclosed
US-5641807-A Method for the treatment of depression ASTRA AKTIEBOLAG (SE) 1997-06-24 US disclosed
US-5639772-A Chroman derivatives ASTRA AKTIEBOLAG (SE) 1997-06-17 US disclosed
US-5639784-A ADMINISTERING 3-AMINO-5-CARBAMOYL-CHROMENES AND DERIVATIVES ASTRA AKTIEBOLAG (SE) 1997-06-17 US disclosed
US-5500425-A Chroman derivatives and a method of treating 5-HT mediated disorders AKTIEBOLAGET ASTRA (SE) 1996-03-19 US disclosed
US-5420151-A Chroman derivatives AKTIEBOLAGET ASTRA (SE) 1995-05-30 US disclosed