SCHEMBL8824809

SCHEMBL8824809

CC(C)(C)OC(=O)n1cc(N)nc1-c1cccc([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
PKM P14618 2/20 0.49
MAPT P10636 7/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
RAB9A P51151 3/20 0.45
NR3C2 P08235 1/20 0.44
LMNA P02545 2/20 0.43
MAPK1 P28482 1/20 0.42
GFER P55789 1/20 0.41
NPC1 O15118 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PTGS2 P35354 1/20 0.41
ALOX5 P09917 1/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29796135 0.80 ALDH1A1 (0.48) ALDH1A1PKMMAPTMEN1KMT2A
SCHEMBL23213140 0.80 ALDH1A1 (0.48) ALDH1A1PKMMAPTMEN1KMT2A
SCHEMBL4606178 0.78 ALDH1A1 (0.57) ALDH1A1PKMMAPTMEN1KMT2A
SCHEMBL4717161 0.76 HSP90AA1 (0.46) ALDH1A1PKMMAPTMEN1KMT2A
SCHEMBL1019778 0.74 F2 (0.45) ALDH1A1PKMMAPTMEN1KMT2A
SCHEMBL20501018 0.74 ALDH1A1 (0.44) ALDH1A1PKMMAPTMEN1KMT2A
SCHEMBL13426427 0.73 PDE4B (0.47) ALDH1A1PKMMAPTRAB9ANR3C2
SCHEMBL31226734 0.73 ALDH1A1 (0.45) ALDH1A1PKMMAPTMEN1KMT2A
SCHEMBL21296822 0.72 ALDH1A1 (0.44) ALDH1A1PKMMAPTRAB9ANR3C2
SCHEMBL29938392 0.72 ALDH1A1 (0.44) ALDH1A1PKMMAPTRAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681833-A ADMINSTERING FOR TREATMENT OF PEPTIC ULCER MERCK, SHARP & DOHME LTD. (GB) 1997-10-28 US disclosed
WO-1993019052-A1 3-UREIDO SUBSTITUTED BENZODIAZEPIN-2-ONES HAVING CHOLECYSTOKININ AND/OR GASTRIN ANTAGONISTIC ACTIVITY AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-09-30 WO disclosed