SCHEMBL8825974

SCHEMBL8825974

O=C(O)C1C(C(=O)N2CCCC(c3ccccc3)C2)C(C(=O)O)C1C(=O)N1CCCC(c2ccccc2)C1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
LMNA P02545 2/20 0.53
HPGD P15428 2/20 0.53
HIF1A Q16665 1/20 0.53
HSD11B1 P28845 2/20 0.52
RAB9A P51151 5/20 0.50
NPC1 O15118 4/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
MAPT P10636 3/20 0.50
POLB P06746 2/20 0.50
TSHR P16473 1/20 0.50
TP53 P04637 1/20 0.50
RECQL P46063 1/20 0.50
PROKR1 Q8TCW9 1/20 0.48
ATM Q13315 1/20 0.48
DRD2 P14416 1/20 0.47
DRD1 P21728 1/20 0.47
DRD4 P21917 1/20 0.47
DRD5 P21918 1/20 0.47
DRD3 P35462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8825970 1.00 ALDH1A1 (0.56) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL11178698 0.84 ALDH1A1 (0.58) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL3312540 0.82 ALDH1A1 (0.62) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL27878990 0.82 ALDH1A1 (0.62) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL23009741 0.80 ALDH1A1 (0.59) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL21424973 0.80 ALDH1A1 (0.59) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL20738614 0.80 ALDH1A1 (0.60) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL21425067 0.80 ALDH1A1 (0.59) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL20738480 0.80 ALDH1A1 (0.60) ALDH1A1LMNAHPGDHIF1AHSD11B1
SCHEMBL21138878 0.80 ALDH1A1 (0.59) ALDH1A1LMNAHPGDHIF1AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5631401-A Inhibitors of protein farnesyltransferase and squalene synthase ABBOTT LABORATORIES (US) 1997-05-20 US disclosed
WO-1995021815-A1 CYCLOBUTANE DERIVATIVES AND THEIR USE AS INHIBITORS OF PROTEIN FARNESYLTRANSFERASE AND SQUALENE SYNTHASE ABBOTT LABORATORIES (US) 1995-08-17 WO disclosed