SCHEMBL8826280

SCHEMBL8826280

CC(C)N(c1ccccc1-c1ccccc1)C(=O)[C@H]1[C@H](C(=O)O)[C@H](C(=O)N(c2ccccc2-c2ccccc2)C(C)C)[C@H]1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 1/20 0.39
KDM4E B2RXH2 3/20 0.38
PKM P14618 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
EDNRB P24530 2/20 0.37
EDNRA P25101 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 4/20 0.37
FABP3 P05413 2/20 0.37
FABP7 O15540 1/20 0.37
FABP5 Q01469 1/20 0.37
TACR1 P25103 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8496545 1.00 GPR88 (0.39) GPR88KDM4EPKMNPSR1SMN1; SMN2
SCHEMBL8696052 0.84 GPR88 (0.42) GPR88NPSR1SMN1; SMN2EDNRBEDNRA
SCHEMBL31393802 0.81 SMN1; SMN2 (0.41) GPR88KDM4EPKMNPSR1SMN1; SMN2
SCHEMBL8825958 0.80 TACR1 (0.47) GPR88KDM4ESMN1; SMN2EDNRBEDNRA
SCHEMBL24359328 0.71 KMT2A (0.41) KDM4ENPSR1SMN1; SMN2MEN1KMT2A
Biphenyl SCHEMBL5496359 0.69 KMT2A (0.41) GPR88PKMSMN1; SMN2MEN1KMT2A
SCHEMBL20152515 0.68 CDC25B (0.40) KDM4ENPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL10787360 0.68 KMT2A (0.40) GPR88NPSR1SMN1; SMN2MEN1KMT2A
SCHEMBL7450697 0.67 TACR1 (0.49) GPR88KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL8693959 0.67 TACR1 (0.43) GPR88KDM4ENPSR1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5631401-A Inhibitors of protein farnesyltransferase and squalene synthase ABBOTT LABORATORIES (US) 1997-05-20 US disclosed
WO-1995021815-A1 CYCLOBUTANE DERIVATIVES AND THEIR USE AS INHIBITORS OF PROTEIN FARNESYLTRANSFERASE AND SQUALENE SYNTHASE ABBOTT LABORATORIES (US) 1995-08-17 WO disclosed