SCHEMBL8828152

SCHEMBL8828152

CN(CCCNC(=O)C/C=C/c1ccc(-n2ccnc2)cc1)CCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 2/20 0.43
SIGMAR1 Q99720 2/20 0.43
NAPEPLD Q6IQ20 1/20 0.42
TBXAS1 P24557 2/20 0.42
ESR1 P03372 1/20 0.42
MAOB P27338 2/20 0.41
GAA P10253 1/20 0.39
CYP4Z1 Q86W10 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
PORCN Q9H237 1/20 0.38
MLLT1 Q03111 1/20 0.38
ACKR3 P25106 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9158516 0.97 TBXAS1 (0.41) TMEM97SIGMAR1NAPEPLDTBXAS1ESR1
SCHEMBL8828318 0.90 DRD3 (0.44) TBXAS1MAOBGAA
SCHEMBL9156723 0.90 MAOB (0.46) TBXAS1ESR1MAOB
SCHEMBL8828168 0.89 DRD3 (0.45) SIGMAR1
SCHEMBL9159739 0.89 MAOB (0.42) TMEM97SIGMAR1TBXAS1MAOB
SCHEMBL8828202 0.88 DRD3 (0.41) MAOBGAA
SCHEMBL9231352 0.88 DRD3 (0.45) TBXAS1MAOBGAA
SCHEMBL9158719 0.87 DRD3 (0.46)
Hydrochloric Acid SCHEMBL6368810 0.87 DRD3 (0.41) MAOBGAA
SCHEMBL9157622 0.86 KCNH2 (0.40) TMEM97SIGMAR1TBXAS1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
US-5177089-A Antiischemic agent, vasodilator EISAI CO., LTD. (JP) 1993-01-05 US disclosed
US-5047417-A Butenoic or propenoic acid derivatives EISAI CO. LTD. (JP) 1991-09-10 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed