SCHEMBL8828401

SCHEMBL8828401

O=C(O)CC=Cc1cc(-n2ccnc2)cs1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 2/20 0.41
ADH5 P11766 5/20 0.39
CYP3A4 P08684 2/20 0.38
BAZ2B Q9UIF8 1/20 0.38
MAOB P27338 3/20 0.36
ENPP2 Q13822 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
CYP11B1 P15538 2/20 0.35
IDO1 P14902 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP11B2 P19099 1/20 0.35
HTT P42858 1/20 0.35
CYP17A1 P05093 1/20 0.35
CYP21A2 P08686 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
MITF O75030 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828392 1.00 TBXAS1 (0.41) TBXAS1ADH5CYP3A4BAZ2BMAOB
SCHEMBL11015694 0.81 TBXAS1 (0.44) TBXAS1ADH5CYP3A4BAZ2BMAOB
SCHEMBL11015693 0.81 TBXAS1 (0.44) TBXAS1ADH5CYP3A4BAZ2BMAOB
SCHEMBL8828266 0.77 MAOB (0.54) TBXAS1ADH5CYP3A4BAZ2BMAOB
SCHEMBL8828261 0.77 MAOB (0.54) TBXAS1ADH5CYP3A4BAZ2BMAOB
SCHEMBL8828222 0.75 IDO1 (0.50) TBXAS1ADH5CYP3A4MAOBCYP11B1
SCHEMBL8828227 0.75 IDO1 (0.50) TBXAS1ADH5CYP3A4MAOBCYP11B1
SCHEMBL10365507 0.75 IDO1 (0.44) ADH5CYP3A4BAZ2BENPP2MKNK1
SCHEMBL8828161 0.75 TBXAS1 (0.39) TBXAS1ADH5CYP3A4BAZ2BMAOB
SCHEMBL8828171 0.75 TBXAS1 (0.39) TBXAS1ADH5CYP3A4BAZ2BMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607953-A ANTIISCHEMIC AGENTS EISAI CO., LTD. (JP) 1997-03-04 US disclosed
EP-0344577-B1 Butenoic or propenoic acid derivatives EISAI CO LTD (JP) 1996-10-09 EP disclosed
US-5382595-A Antiischemic agents EISAI CO., LTD. (JP) 1995-01-17 US disclosed
EP-0344577-A2 Butenoic or propenoic acid derivatives Eisai Co., Ltd. (JP) 1989-12-06 EP disclosed