SCHEMBL8832161

SCHEMBL8832161

COc1ccc(/C=C/C(=O)Oc2ccc([N+](=O)[O-])cc2)cc1N(C)C

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.52
CYP19A1 P11511 1/20 0.52
KRAS P01116 2/20 0.50
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
TLR9 Q9NR96 1/20 0.50
ALDH1A1 P00352 3/20 0.49
KMT2A Q03164 2/20 0.49
KDM4E B2RXH2 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MMP1 P03956 1/20 0.48
APP P05067 1/20 0.48
MAPT P10636 5/20 0.48
GAA P10253 2/20 0.48
LMNA P02545 2/20 0.46
TXNRD1 Q16881 1/20 0.45
TXNRD3 Q86VQ6 1/20 0.45
TXNRD2 Q9NNW7 1/20 0.45
HTT P42858 1/20 0.45
RECQL P46063 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8832165 1.00 PTGS2 (0.52) PTGS2CYP19A1KRASMAOAMAOB
SCHEMBL9523759 0.87 PTGS2 (0.69) PTGS2CYP19A1KRASMAOAMAOB
SCHEMBL9523755 0.87 PTGS2 (0.69) PTGS2CYP19A1KRASMAOAMAOB
SCHEMBL9522624 0.85 CYP19A1 (0.55) PTGS2CYP19A1KRASMAOAMAOB
SCHEMBL9522627 0.85 CYP19A1 (0.55) PTGS2CYP19A1KRASMAOAMAOB
SCHEMBL30839393 0.83 MAPT (0.66) PTGS2CYP19A1MAOAMAOBTLR9
SCHEMBL1597196 0.83 MAPT (0.66) PTGS2CYP19A1MAOAMAOBTLR9
SCHEMBL9478343 0.81 MAOB (0.73) PTGS2KRASMAOAMAOBTLR9
SCHEMBL9478353 0.81 MAOB (0.73) PTGS2KRASMAOAMAOBTLR9
SCHEMBL8832242 0.81 MAPT (0.53) PTGS2CYP19A1ALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670492-A BACTERICIDE, ANTITUMOR AGENT KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-09-23 US disclosed
EP-0702014-A1 DC-89 DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 1996-03-20 EP disclosed