SCHEMBL8836007

SCHEMBL8836007

CCOC(=O)c1c(NCc2ccccc2CC(=O)c2ccccc2)c2c(Cl)cc(Cl)cc2n1C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 5/20 0.43
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
ROCK2 O75116 1/20 0.36
CHEK2 O96017 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KA3 P51812 1/20 0.36
PAK1 Q13153 1/20 0.36
ROCK1 Q13464 1/20 0.36
DYRK1A Q13627 1/20 0.36
PRKD2 Q9BZL6 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
SLC26A6 Q9BXS9 1/20 0.34
NR1H2 P55055 1/20 0.34
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8836014 0.89 MDM2 (0.46) MDM2KDM4EHPGDROCK2CHEK2
SCHEMBL8540513 0.88 MDM2 (0.48) MDM2KDM4EHPGDLMNASMN1; SMN2
SCHEMBL8538967 0.86 MDM2 (0.44) MDM2KDM4EHPGDLMNASMN1; SMN2
SCHEMBL8541910 0.85 MDM2 (0.43) MDM2KDM4EHPGDNR1H2CRHBP
SCHEMBL8540675 0.83 MDM2 (0.46) MDM2KDM4EHPGDLMNASMN1; SMN2
SCHEMBL8541107 0.82 MDM2 (0.47) MDM2LMNASMN1; SMN2CRHBPCRHR2
SCHEMBL8541912 0.82 MDM2 (0.45) MDM2KDM4EHPGDLMNASMN1; SMN2
SCHEMBL8541135 0.82 MDM2 (0.43) MDM2KDM4EHPGDL3MBTL1NR1H2
SCHEMBL8540708 0.81 MDM2 (0.42) MDM2HPGDLMNASMN1; SMN2CYP1A2
SCHEMBL8541127 0.81 MDM2 (0.44) MDM2KDM4EHPGDLMNANR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703107-A CENTRAL NERVOUS SYSTEM DISORDERS; ANALGESICS; ANTIEPILEPTIC AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-12-30 US disclosed