SCHEMBL8836192

SCHEMBL8836192

O=C(c1cc2ccccc2o1)N1CCN(C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)[C@H](Cc2ccccc2)C1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.58
CA1 P00915 10/20 0.52
CA2 P00918 10/20 0.52
CA4 P22748 10/20 0.52
CA9 Q16790 10/20 0.52
ALDH1A1 P00352 1/20 0.51
GRIN2B Q13224 1/20 0.47
HRH4 Q9H3N8 1/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8479813 0.84 TACR1 (0.58) TACR1CA1CA2CA4CA9
SCHEMBL8480544 0.83 TACR1 (0.63) TACR1CA1CA2CA4CA9
SCHEMBL8475935 0.83 CA1 (0.65) TACR1CA1CA2CA4CA9
SCHEMBL8480058 0.82 CA1 (0.66) TACR1CA1CA2CA4CA9
SCHEMBL8481073 0.81 TACR1 (0.61) TACR1CA1CA2CA4CA9
SCHEMBL6100617 0.81 TACR1 (0.61) TACR1CA1CA2CA4CA9
SCHEMBL9241572 0.80 TACR1 (0.58) TACR1CA1CA2CA4CA9
SCHEMBL9241579 0.80 TACR1 (0.58) TACR1CA1CA2CA4CA9
SCHEMBL6099419 0.80 TACR1 (0.43) TACR1CA1CA2CA4CA9
SCHEMBL8476168 0.80 TACR1 (0.60) TACR1CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670505-A TACHYKIKIN ANTAGONIST FOR RESPIRATORY DISEASES, OPHTHALMIC DISEASES AND ANTIINFLAMMATORY AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-23 US disclosed
US-5670540-A NUTRITIONAL SUPPLEMENT SCOTIA HOLDINGS PLC (GB) 1997-09-23 US disclosed
EP-0655442-A1 Piperazine derivatives as Tachykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-05-31 EP disclosed