SCHEMBL8842653

SCHEMBL8842653

COc1cc(C2=NCCN2)ccc1-c1ccnc(-c2ccc(C3=NCCN3)cc2)n1

nearest known ligand 0.60

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.54
NISCH Q9Y2I1 5/20 0.51
S1PR1 P21453 1/20 0.47
PDCD1LG2 Q9BQ51 5/20 0.47
CD274 Q9NZQ7 5/20 0.47
MAOA P21397 2/20 0.44
PTGIR P43119 1/20 0.44
KDM4E B2RXH2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8894710 0.78 LMNA (0.56) MAOBNISCHMAOA
SCHEMBL9575182 0.76 MAOB (0.69) MAOBNISCHPTGIRKDM4E
SCHEMBL29014990 0.74 NPC1 (0.60) KDM4E
SCHEMBL30450715 0.74 NPC1 (0.60) KDM4E
SCHEMBL13175784 0.74 NISCH (0.60) MAOBNISCHPTGIRKDM4E
SCHEMBL30980862 0.73 NISCH (0.55) MAOBNISCHPDCD1LG2CD274
SCHEMBL8842460 0.73 MEN1 (0.50) KDM4E
Hydrochloric Acid SCHEMBL8842474 0.73 NISCH (0.64) MAOBNISCHMAOA
SCHEMBL8842604 0.73 CYP1A1 (0.49)
SCHEMBL27650161 0.72 MAOB (0.49) MAOBNISCHPDCD1LG2CD274MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686456-A DIARYLPYRIMIDINES THE UNIVERSITY OF NORTH CAROLINA (US) 1997-11-11 US disclosed
US-5627184-A BACTERICIDES OF PYRIMIDINE DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-05-06 US disclosed
US-5622955-A ADMINISTERING 2,4-BIS-/4-GUANYLPHENYL/-PYRIMIDINE OR DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-04-22 US disclosed
US-5606058-A HAVING REDUCED SIDE EFFECTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-02-25 US disclosed
US-5521189-A PYRIMIDINE COMPOUNDS AS ANTIPROTOZOA AGENTS THE UNIVERSITY OF NC AT CH (US) 1996-05-28 US disclosed