SCHEMBL8842886

SCHEMBL8842886

CC(CC(=O)O)NC(=O)c1cc(I)ccc1N(C)c1ccc2ccccc2c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.36
EGLN2 Q96KS0 3/20 0.36
EGLN1 Q9GZT9 3/20 0.36
KCNB1 Q14721 1/20 0.35
KCNB2 Q92953 1/20 0.35
PYGL P06737 2/20 0.35
POLR1A O95602 1/20 0.35
GAA P10253 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PDPK1 O15530 1/20 0.34
MAOB P27338 1/20 0.34
NPC1 O15118 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8837019 0.90 TACR3 (0.36) POLR1AGAARAB9ASMN1; SMN2KMT2A
SCHEMBL8842974 0.89 CYP26A1 (0.46) KMT2A
SCHEMBL7329795 0.83 TACR3 (0.48) NPC1KMT2AMEN1
SCHEMBL7564581 0.83 TACR3 (0.48) NPC1KMT2AMEN1
SCHEMBL7333801 0.75 GAA (0.39) GAASMN1; SMN2ALDH1A1
SCHEMBL7325460 0.72 PTPRC (0.38) EGLN1PYGLGAAKMT2AMEN1
SCHEMBL9829253 0.68 PLK1 (0.55) RAB9ASMN1; SMN2NPC1KMT2AMEN1
SCHEMBL1114971 0.67 TTR (0.40) EGLN2EGLN1KMT2AMEN1
SCHEMBL18799916 0.66 HTT (0.41) RAB9ANPC1ALDH1A1
SCHEMBL1114965 0.66 KDM4E (0.62) GAARAB9ASMN1; SMN2NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663166-A ANTICOAGULANTS OF 1,4-BENZODIAZEPINE-2,5-DIONE AND 2-BENZOAZEPINE-1,4-DIONE DERIVATIVES; PREVENTS FIBRINOGEN BINDING NECESSARY FOR PLATELET AGGREGATION; SIDE EFFECT REDUCTION, E.G. EXCESSIVE BLEEDING GENENTECH, INC. (US) 1997-09-02 US disclosed