SCHEMBL8842974

SCHEMBL8842974

CN(c1ccc2ccccc2c1)c1ccc(I)cc1C(=O)NC(CC(=O)O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 10/20 0.46
CTSA P10619 2/20 0.41
TACR3 P29371 2/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
UTS2R Q9UKP6 4/20 0.38
MMP12 P39900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329795 0.92 TACR3 (0.48) CYP26A1CTSATACR3KMT2ATDP1
SCHEMBL7564581 0.92 TACR3 (0.48) CYP26A1CTSATACR3KMT2ATDP1
SCHEMBL8842886 0.89 CASP1 (0.36) KMT2A
SCHEMBL8837019 0.81 TACR3 (0.36) TACR3KMT2AUTS2R
SCHEMBL7333801 0.73 GAA (0.39)
SCHEMBL5926568 0.71 CTSA (0.42) CYP26A1CTSAKMT2AMMP12
SCHEMBL5425777 0.70 CYP26A1 (0.52) CYP26A1CTSATACR3KMT2ATDP1
SCHEMBL5926664 0.69 CTSA (0.53) CYP26A1CTSATACR3MMP12
SCHEMBL7335381 0.68 ALDH1A1 (0.49) CYP26A1TACR3KMT2A
SCHEMBL7332776 0.67 ALDH1A1 (0.44) CYP26A1TACR3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663166-A ANTICOAGULANTS OF 1,4-BENZODIAZEPINE-2,5-DIONE AND 2-BENZOAZEPINE-1,4-DIONE DERIVATIVES; PREVENTS FIBRINOGEN BINDING NECESSARY FOR PLATELET AGGREGATION; SIDE EFFECT REDUCTION, E.G. EXCESSIVE BLEEDING GENENTECH, INC. (US) 1997-09-02 US disclosed